SCHEMBL18852736

SCHEMBL18852736

CCc1cnc2c(ccn2C(C)(C)C)c1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP1A2 P05177 2/20 0.32
KDM4E B2RXH2 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
ATM Q13315 1/20 0.32
CYP2A6 P11509 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21167296 0.80 APP (0.36)
SCHEMBL12524710 0.78 CHRNA7 (0.41) PARP1MAPTCYP1A2CYP2D6CYP2A6
SCHEMBL26014245 0.77 IRAK4 (0.35) MAPTCYP1A2KDM4ECYP3A4CYP2D6
SCHEMBL26596996 0.77 PIK3CB (0.34) MAPTKDM4E
SCHEMBL18125589 0.77 KCNH2 (0.33) MEN1KMT2ACYP1A2KDM4ECYP3A4
SCHEMBL26433112 0.76 CDK4 (0.33)
SCHEMBL22761968 0.74 GRIN2B (0.40) MEN1KMT2ANPC1TP53MAPT
SCHEMBL26433102 0.73 ABL1 (0.33) MAPT
SCHEMBL21704228 0.73 PARP1 (0.35) PARP1CYP1A2CYP2A6
SCHEMBL23937881 0.72 PARP1 (0.37) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9650379-B2 Azaindole derivatives as selective histone deacetylase (HDAC) inhibitors and pharmaceutical compositions comprising the same CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2017-05-16 US disclosed