SCHEMBL18857014

SCHEMBL18857014

Brc1ccc2c(ccn2CI)c1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.58
HTR2C P28335 2/20 0.58
HTR7 P34969 2/20 0.49
NTSR1 P30989 1/20 0.44
KRAS P01116 7/20 0.41
SLC6A2 P23975 2/20 0.40
ROCK1 Q13464 1/20 0.40
MCL1 Q07820 1/20 0.38
FABP3 P05413 1/20 0.37
FABP2 P12104 1/20 0.37
FABP4 P15090 1/20 0.37
FABP5 Q01469 1/20 0.37
AR P10275 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3478164 0.81 HTR2A (0.63) HTR2AHTR2CHTR7NTSR1KRAS
SCHEMBL18301155 0.80 HTR2A (0.54) HTR2AHTR2CHTR7NTSR1KRAS
SCHEMBL3046803 0.78 HTR2A (0.55) HTR2AHTR2CHTR7NTSR1KRAS
SCHEMBL27976945 0.78 HTR2A (0.55) HTR2AHTR2CHTR7NTSR1
SCHEMBL21941497 0.78 HTR2A (0.59) HTR2AHTR2CHTR7NTSR1KRAS
SCHEMBL14061899 0.78 HTR2A (0.59) HTR2AHTR2CHTR7NTSR1KRAS
SCHEMBL4944251 0.78 HTR2C (0.68) HTR2AHTR2CHTR7NTSR1KRAS
SCHEMBL18856961 0.77 HTR2A (0.58) HTR2AHTR2CKRASSLC6A2
SCHEMBL18856956 0.77 HTR2C (0.58) HTR2AHTR2CFABP4AR
SCHEMBL2382637 0.77 HTR2A (0.54) HTR2AHTR2CHTR7NTSR1KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017082924-A1 PEPTIDE AND PEPTIDE MIMETIC BINDING ANTAGONISTS OF POLO-LIKE KINASE 1 POLO BOX DOMAIN AND METHODS OF USE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2017-05-18 WO disclosed