SCHEMBL18870546

SCHEMBL18870546

CC(C)(C)OC(=O)N1CCCC[C@H]1c1ncc(-c2ccc(B3OC(C)(C)C(C)(C)O3)cc2)[nH]1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.46
CYP3A4 P08684 3/20 0.45
CYP2C9 P11712 3/20 0.45
NR1I2 O75469 1/20 0.45
ABCB11 O95342 1/20 0.45
OPRK1 P41145 1/20 0.45
KCNH2 Q12809 1/20 0.45
PRCP P42785 5/20 0.44
HPGDS O60760 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 1/20 0.43
OPRM1 P35372 2/20 0.41
OPRD1 P41143 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL204943 0.97 CYP3A4 (0.48) USP30CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL2706319 0.97 CYP3A4 (0.48) USP30CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL203309 0.97 CYP3A4 (0.48) USP30CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL15083853 0.96 CYP3A4 (0.49) USP30CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL19488538 0.91 PRCP (0.47) USP30PRCPHPGDSOPRM1OPRD1
SCHEMBL205276 0.90 CYP3A4 (0.46) USP30CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL205250 0.90 PRCP (0.46) USP30CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL2707681 0.90 PRCP (0.46) USP30CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL2707737 0.90 CYP3A4 (0.46) USP30CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL204202 0.90 PRCP (0.45) USP30CYP3A4CYP2C9NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2601188-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-10-18 EP disclosed
EP-2900656-B1 SPIRO RING COMPOUNDS AS HEPATITIS C VIRUS (HCV) INHIBITORS SUNSHINE LAKE PHARMA CO LTD (CN) 2017-05-17 EP disclosed