SCHEMBL18879484

SCHEMBL18879484

CC1(C)CC(N)CN(c2ccc(C#N)c3ncccc23)C1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 12/20 0.60
TLR9 Q9NR96 13/20 0.48
TLR7 Q9NYK1 13/20 0.48
AR P10275 1/20 0.34
NSD2 O96028 1/20 0.34
HRH1 P35367 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
RPS6KB1 P23443 1/20 0.34
ELANE P08246 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18879482 1.00 TLR8 (0.60) TLR8TLR9TLR7ARNSD2
Hydrochloric Acid SCHEMBL17840531 0.99 TLR8 (0.59) TLR8TLR9TLR7ARNSD2
Hydrochloric Acid SCHEMBL17840529 0.99 TLR8 (0.59) TLR8TLR9TLR7ARNSD2
SCHEMBL19000090 0.87 TLR8 (0.63) TLR8TLR9TLR7ARNSD2
SCHEMBL23855164 0.87 TLR8 (0.63) TLR8TLR9TLR7ARNSD2
SCHEMBL18980745 0.86 TLR8 (0.43) TLR8TLR9TLR7
SCHEMBL18980747 0.86 TLR8 (0.43) TLR8TLR9TLR7
Hydrochloric Acid SCHEMBL18980484 0.86 TLR8 (0.62) TLR8TLR9TLR7ARNSD2
Hydrochloric Acid SCHEMBL18980842 0.85 TLR8 (0.43) TLR8TLR9TLR7
SCHEMBL16653627 0.81 TLR8 (0.45) TLR8TLR9TLR7ARRPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057948-B1 SELECTIVELY SUBSTITUTED QUINOLINE DERIVATIVES EISAI R&D MAN CO LTD (JP) 2018-03-14 EP claimed
US-9663486-B2 Selectively substituted quinoline compounds EISAI R&D MANAGEMENT CO., LTD. (JP) 2017-05-30 US claimed