SCHEMBL18895809

SCHEMBL18895809

C/N=C/c1cc(-c2ccc(F)cc2)c2ccc(CN3C(=O)COC3=O)cc2n1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 20/20 0.67
NR1I2 O75469 2/20 0.49
KCNH2 Q12809 2/20 0.49
GRM6 O15303 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19336356 0.88 GRM2 (0.70) GRM2NR1I2KCNH2GRM6
SCHEMBL18895801 0.88 GRM2 (0.64) GRM2NR1I2KCNH2GRM6
SCHEMBL18799975 0.84 GRM2 (0.68) GRM2NR1I2KCNH2GRM6
SCHEMBL18799979 0.83 GRM2 (0.68) GRM2NR1I2KCNH2GRM6
SCHEMBL19336358 0.81 GRM2 (0.72) GRM2NR1I2KCNH2GRM6
SCHEMBL18895813 0.81 GRM2 (0.67) GRM2NR1I2KCNH2GRM6
SCHEMBL14933124 0.80 GRM2 (1.00) GRM2NR1I2KCNH2GRM6
SCHEMBL19336334 0.75 GRM2 (0.68) GRM2NR1I2KCNH2GRM6
SCHEMBL19336363 0.73 GRM2 (0.70) GRM2NR1I2KCNH2GRM6
SCHEMBL19336347 0.72 GRM2 (0.71) GRM2NR1I2KCNH2GRM6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9663506-B2 Quinoline carboxamide and quinoline carbonitrile derivatives as mGluR2-negative allosteric modulators, compositions, and their use MERCK SHARP & DOHME CORP. (US) 2017-05-30 US disclosed