SCHEMBL18895993

SCHEMBL18895993

CN(C)C(=O)COc1ccc2c(c1)C(=CCCN1CCC(N=O)(c3ccc(Cl)cc3)CC1)c1cccnc1CO2

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.54
CHRM2 P08172 1/20 0.48
CCR5 P51681 1/20 0.48
HRH1 P35367 6/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
HTR2B P41595 1/20 0.31
S1PR5 Q9H228 2/20 0.31
LMNA P02545 1/20 0.30
PDK2 Q15119 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15478358 0.92 CCR1 (0.54) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL10288256 0.91 CCR1 (0.57) CCR1CHRM2CCR5HRH1ADRA1A
SCHEMBL12121719 0.88 CCR1 (0.54) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL10288250 0.86 CCR1 (0.53) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL14420032 0.86 CCR1 (0.53) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL10287596 0.85 CCR1 (0.52) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL15478344 0.85 CCR1 (0.59) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL14579621 0.85 CCR1 (0.54) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL15478347 0.85 CCR1 (0.51) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL15478312 0.84 CCR1 (0.48) CCR1CHRM2CCR5HRH1ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9663537-B2 Chemokine receptor antagonists and methods of use MILLENNIUM PHARMACEUTICALS, INC. (US) 2017-05-30 US disclosed