SCHEMBL18898643

SCHEMBL18898643

CCc1cnc2[nH]c(=O)n(C(C)C)c2n1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTOR P42345 5/20 0.55
CYP1A2 P05177 1/20 0.50
FYN P06241 1/20 0.36
CDK1 P06493 1/20 0.34
POLB P06746 2/20 0.33
MAPK8 P45983 1/20 0.33
ADORA2B P29275 1/20 0.33
MAP3K11 Q16584 2/20 0.32
IL6 P05231 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
ALDH1A1 P00352 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
CCND2 P30279 1/20 0.31
CCND3 P30281 1/20 0.31
PDE5A O76074 1/20 0.31
PDE6C P51160 1/20 0.31
PDE4D Q08499 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL976625 0.87 CYP1A2 (0.66) MTORCYP1A2FYNMAP3K11PDE4D
SCHEMBL975430 0.83 FYN (0.54) MTORCYP1A2FYN
SCHEMBL975431 0.83 FYN (0.54) MTORCYP1A2FYN
SCHEMBL19200211 0.80 MTOR (0.53) MTORCYP1A2FYNCDK1POLB
SCHEMBL17807738 0.79 MTOR (0.58) MTORCYP1A2FYNPOLBMAPK8
SCHEMBL481934 0.79 MTOR (0.58) MTORCYP1A2FYNCDK1POLB
SCHEMBL24995677 0.77 MTOR (0.55) MTORCYP1A2FYNPOLBMAPK8
SCHEMBL975519 0.77 MTOR (0.55) MTORCYP1A2FYNPOLBMAPK8
SCHEMBL977817 0.75 CYP1A2 (0.55) MTORCYP1A2PDE4D
SCHEMBL19200146 0.75 POLB (0.44) MTORCDK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9663520-B2 Bicyclic bromodomain inhibitors ZENITH EPIGENETICS LTD. (CA) 2017-05-30 US disclosed