SCHEMBL18901347

SCHEMBL18901347

CN(CC(=O)O)Cc1ccc(-c2noc(-c3ccc(-c4ccccc4C(C)(F)F)c(I)c3)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 16/20 0.48
HDAC4 P56524 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC7 Q8WUI4 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HDAC5 Q9UQL6 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC9 Q9UKV0 1/20 0.41
S1PR3 Q99500 3/20 0.40
S1PR5 Q9H228 1/20 0.40
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18901348 0.90 S1PR1 (0.54) S1PR1HDAC4HDAC1HDAC7HDAC6
SCHEMBL18901332 0.87 S1PR1 (0.54) S1PR1HDAC4HDAC1HDAC7HDAC6
SCHEMBL557673 0.84 S1PR1 (0.59) S1PR1HDAC4HDAC1HDAC7HDAC6
SCHEMBL10170274 0.83 S1PR1 (0.52) S1PR1HDAC4HDAC1HDAC7HDAC6
SCHEMBL18901333 0.83 S1PR1 (0.53) S1PR1HDAC4HDAC1HDAC7HDAC6
SCHEMBL18901335 0.83 S1PR1 (0.53) S1PR1HDAC4HDAC1HDAC7HDAC6
SCHEMBL558227 0.82 S1PR1 (0.68) S1PR1S1PR3S1PR5
SCHEMBL558155 0.82 S1PR1 (0.61) S1PR1S1PR3S1PR5
SCHEMBL558902 0.82 S1PR1 (0.58) S1PR1S1PR3S1PR5
SCHEMBL18901343 0.82 S1PR1 (0.52) S1PR1S1PR3S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414342-B1 OXADIAZOLE DERIVATIVES MERCK SERONO SA (CH) 2017-05-31 EP disclosed