SCHEMBL18912239

SCHEMBL18912239

CO[C@H]1CCN(c2cccc(-c3nc(-n4nc(C)cc4C)nc(N)c3C#N)n2)C1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.52
ADORA1 P30542 11/20 0.52
TSPO P30536 1/20 0.52
GPR183 P32249 1/20 0.52
SIGMAR1 Q99720 1/20 0.52
GPR35 Q9HC97 1/20 0.52
CYP3A4 P08684 1/20 0.49
KCNH2 Q12809 1/20 0.38
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
ALOX15 P16050 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PIM1 P11309 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18912381 1.00 ADORA2A (0.52) ADORA2AADORA1TSPOGPR183SIGMAR1
SCHEMBL18912275 1.00 ADORA2A (0.52) ADORA2AADORA1TSPOGPR183SIGMAR1
SCHEMBL30252565 1.00 ADORA2A (0.52) ADORA2AADORA1TSPOGPR183SIGMAR1
SCHEMBL18912230 0.95 ADORA2A (0.57) ADORA2AADORA1TSPOGPR183SIGMAR1
SCHEMBL18893656 0.88 ADORA2A (0.51) ADORA2AADORA1TSPOGPR183SIGMAR1
SCHEMBL18912279 0.88 ADORA2A (0.51) ADORA2AADORA1TSPOGPR183SIGMAR1
SCHEMBL18893683 0.88 ADORA2A (0.51) ADORA2AADORA1TSPOGPR183SIGMAR1
SCHEMBL20911174 0.87 ADORA2A (0.47) ADORA2AADORA1TSPOGPR183SIGMAR1
SCHEMBL28995967 0.87 ADORA2A (0.47) ADORA2AADORA1TSPOGPR183SIGMAR1
SCHEMBL18912277 0.86 ADORA2A (0.57) ADORA2AADORA1TSPOGPR183SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017088755-A1 AMINOPYRIMIDINE HETEROCYCLIC COMPOUND WITH ADENOSINE RECEPTOR ANTAGONISTIC ACTIVITY Suzhou Yunxuan Yiyao Keji Youxian Gongsi (CN) 2017-06-01 WO disclosed