SCHEMBL18928331

SCHEMBL18928331

Cc1c(-c2c(C)c3c(c(C)c2CC(=O)O)CC(=O)N(C2CCOCC2)C3)cc(F)c2c1CCCO2

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.36
PDE4A P27815 3/20 0.36
CREBBP Q92793 3/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18928355 0.95 NR1I2 (0.36) NR1I2PDE4ACREBBP
SCHEMBL18928380 0.93 PDE4A (0.36) NR1I2PDE4APTGDR2
SCHEMBL18928319 0.92 NR1I2 (0.34) NR1I2PDE4A
SCHEMBL18928496 0.89 NR1I2 (0.34) NR1I2PDE4A
SCHEMBL18928003 0.89 NR1I2 (0.33) NR1I2PDE4A
SCHEMBL18928342 0.88 NR1I2 (0.37) NR1I2PDE4APTGDR2
SCHEMBL18928563 0.87 NR1I2 (0.35) NR1I2PDE4A
SCHEMBL18928500 0.86 NR1I2 (0.34) NR1I2PDE4A
SCHEMBL18928374 0.86 NR1I2 (0.34) NR1I2PDE4A
SCHEMBL18929018 0.85 PDE4A (0.37) NR1I2PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017093938-A1 TETRAHYDROISOQUINOLINE DERIVATIVES VIIV HEALTHCARE UK LIMITED (GB) 2017-06-08 WO disclosed