SCHEMBL18933467

SCHEMBL18933467

CN(C/C=C/C(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)c(C#N)cnc2cc1OC1CCOC1)CCO

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.69
ERBB2 P04626 12/20 0.68
GAK O14976 3/20 0.66
ABL1 P00519 3/20 0.66
LCK P06239 3/20 0.66
MET P08581 3/20 0.66
PHKG2 P15735 3/20 0.66
BLK P51451 3/20 0.66
ERBB4 Q15303 3/20 0.66
EPHA6 Q9UF33 3/20 0.66
CIT O14578 2/20 0.66
STK10 O94804 2/20 0.66
LYN P07948 2/20 0.66
HCK P08631 2/20 0.66
SRC P12931 2/20 0.66
AXL P30530 2/20 0.66
FLT3 P36888 2/20 0.66
TXK P42681 2/20 0.66
FRK P42685 2/20 0.66
CSNK1E P49674 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15222034 1.00 EGFR (0.69) EGFRERBB2GAKABL1LCK
SCHEMBL15222046 0.95 EGFR (0.66) EGFRERBB2GAKABL1LCK
SCHEMBL18933495 0.95 EGFR (0.66) EGFRERBB2GAKABL1LCK
SCHEMBL14855126 0.94 EGFR (0.69) EGFRERBB2GAKABL1LCK
SCHEMBL18933551 0.94 EGFR (0.69) EGFRERBB2GAKABL1LCK
SCHEMBL21573267 0.94 EGFR (0.70) EGFRERBB2GAKABL1LCK
SCHEMBL14864917 0.94 EGFR (0.70) EGFRERBB2GAKABL1LCK
SCHEMBL14854646 0.93 EGFR (0.78) EGFRERBB2GAKABL1LCK
SCHEMBL14854644 0.93 EGFR (0.78) EGFRERBB2GAKABL1LCK
SCHEMBL14854648 0.93 EGFR (0.78) EGFRERBB2GAKABL1LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3222620-B1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO LTD (CN) 2019-11-20 EP disclosed
EP-3222620-A1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO., LTD. (CN) 2017-09-27 EP disclosed
EP-2581372-B1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO LTD (CN) 2017-06-07 EP disclosed