SCHEMBL18941908

SCHEMBL18941908

Fc1ccc(-c2cnc3[nH]cc(-c4ccnc(NC5CCCC5)n4)c3c2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 10/20 0.66
CCNA2 P20248 8/20 0.66
CDK9 P50750 8/20 0.66
CCNT1 O60563 7/20 0.66
RET P07949 7/20 0.64
CDK1 P06493 5/20 0.62
CDC7 O00311 4/20 0.62
MAP4K4 O95819 4/20 0.62
PRKACA P17612 4/20 0.62
HIPK2 Q9H2X6 4/20 0.62
MKNK2 Q9HBH9 4/20 0.62
IRAK4 Q9NWZ3 4/20 0.62
CCNB1 P14635 3/20 0.62
JAK2 O60674 3/20 0.62
INSR P06213 3/20 0.62
PIM1 P11309 3/20 0.62
FLT3 P36888 3/20 0.62
GSK3B P49841 3/20 0.62
JAK3 P52333 3/20 0.62
ITK Q08881 3/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18941192 0.99 CDK2 (0.64) CDK2CCNA2CDK9CCNT1RET
SCHEMBL18941888 0.96 CCNT1 (0.68) CDK2CCNA2CDK9CCNT1RET
SCHEMBL18941879 0.91 CDK2 (0.66) CDK2CCNA2CDK9CCNT1RET
SCHEMBL18941254 0.90 CDK2 (0.64) CDK2CCNA2CDK9CCNT1RET
SCHEMBL18941853 0.90 CDK2 (0.66) CDK2CCNA2CDK9CCNT1RET
SCHEMBL18941027 0.90 RET (0.64) CDK2CCNA2CDK9CCNT1RET
SCHEMBL18941892 0.89 CDK2 (0.67) CDK2CCNA2CDK9CCNT1RET
SCHEMBL18941279 0.89 CDK1 (0.64) CDK2CCNA2CDK9CCNT1RET
SCHEMBL18941035 0.89 CDK2 (0.64) CDK2CCNA2CDK9CCNT1RET
SCHEMBL18941300 0.88 CDK2 (0.66) CDK2CCNA2CDK9CCNT1RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3383875-B1 3-PYRIMIDINYL PYRROLO [2,3-B] PYRIDINE AS ANTICANCER AGENTS AND THE PROCESS FOR THE PREPARATION THEREOF COUNCIL SCIENT IND RES (IN) 2022-02-09 EP disclosed
WO-2017094026-A1 3-PYRIMIDINYL PYRROLO [2,3-B] PYRIDINE AS NEW ANTICANCER AGENTS AND THE PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2017-06-08 WO disclosed