SCHEMBL18944286

SCHEMBL18944286

CN1CC2=C(Nc3ccccc3NC2=O)N1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.41
CREBBP Q92793 3/20 0.41
LRRK2 Q5S007 3/20 0.39
ACVR1 Q04771 2/20 0.39
PDGFRA P16234 1/20 0.39
FER P16591 1/20 0.39
LTK P29376 1/20 0.39
CDK8 P49336 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
ROS1 P08922 1/20 0.36
CDK5 Q00535 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
CSNK1G1 Q9HCP0 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GLA P06280 1/20 0.34
GSK3B P49841 1/20 0.34
NPC1 O15118 2/20 0.33
BRPF1 P55201 2/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5697347 0.66 ACVR1 (0.67) CREBBPLRRK2ACVR1PDGFRAFER
SCHEMBL8590983 0.65 ACVR1 (0.44) BRD4CREBBPLRRK2ACVR1PDGFRA
SCHEMBL12220595 0.62 ACVR1 (0.50) BRD4CREBBPLRRK2ACVR1PDGFRA
SCHEMBL11168286 0.62 ACVR1 (0.41) BRD4CREBBPLRRK2ACVR1PDGFRA
SCHEMBL4896663 0.60 ACVR1 (0.42) LRRK2ACVR1PDGFRAFERLTK
SCHEMBL9793275 0.60 ACVR1 (0.47) BRD4CREBBPLRRK2ACVR1PDGFRA
SCHEMBL11180043 0.59 CREBBP (0.39) BRD4CREBBPLRRK2ACVR1PDGFRA
SCHEMBL12242976 0.59 ACVR1 (0.56) CREBBPLRRK2ACVR1PDGFRAFER
SCHEMBL677636 0.58 BRD4 (1.00) BRD4CREBBPNPC1MAPK13MAPK12
SCHEMBL23484522 0.58 CREBBP (0.47) BRD4CREBBPLRRK2ACVR1PDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781661-B1 VASOPRESSIN V1A ANTAGONISTS VANTIA LTD (GB) 2017-06-07 EP disclosed