SCHEMBL189560

SCHEMBL189560

O=[N+]([O-])c1cccc(CBr)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.67
LMNA P02545 2/20 0.61
CYP1A2 P05177 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C9 P11712 1/20 0.61
CYP2C19 P33261 1/20 0.61
ALDH1A1 P00352 4/20 0.58
PYCR1 P32322 1/20 0.54
ACHE P22303 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
ALOX15 P16050 1/20 0.52
KMT2A Q03164 2/20 0.50
POLB P06746 1/20 0.50
MEN1 O00255 1/20 0.50
MAPT P10636 1/20 0.50
HSP90AA1 P07900 1/20 0.50
GAA P10253 1/20 0.48
HTT P42858 1/20 0.48
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833623 1.00 TSHR (0.67) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL2928940 0.89 TSHR (0.54) TSHRLMNACYP1A2CYP2D6CYP2C9
Dinitrophenylene SCHEMBL27831167 0.89 TSHR (0.63) TSHRLMNACYP1A2CYP2D6CYP2C9
Formic Acid Methyl Ester SCHEMBL28356814 0.88 CYP2C19 (0.55) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL28638417 0.86 TSHR (0.51) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL18347106 0.85 TSHR (0.62) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL850312 0.85 TSHR (0.62) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL29531585 0.85 TSHR (0.62) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL10918542 0.83 TSHR (0.71) TSHRLMNACYP1A2CYP2D6CYP2C9
Bromide SCHEMBL20258220 0.83 TSHR (0.61) TSHRLMNACYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2231 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116375643-B Deaconitine derivative and preparation method and application thereof 中国人民解放军海军军医大学 2025-04-01 CN claimed
CN-119569808-A Method for modifying C-21 position structure of fusidic acid 浙江工业大学 2025-03-07 CN claimed
CN-118554122-A PI nanofiber composite membrane with lithium dendrite inhibition function and preparation and application thereof 河北科技大学 2024-08-27 CN claimed
CN-116496335-B Modified nucleotide and application thereof 中国药科大学 2024-03-08 CN claimed
CN-116496335-A Modified nucleotide and application thereof 中国药科大学 2023-07-28 CN claimed
CN-116375643-A Deaconitine derivative and preparation method and application thereof 中国人民解放军海军军医大学 2023-07-04 CN claimed
CN-111004228-B GSK-3 beta/ChE double inhibitor and preparation method and application thereof 中国药科大学 2023-05-23 CN claimed
US-20210214372-A1 SMALL MOLECULE ANTAGONIST COMPOUND TAC5 SERIES HAVING TOLL-LIKE RECEPTOR 3/7/8/9 INHIBITORY FUNCTION AJOU UNIVERSITY INDUSTRY-ACADEMIC COOPERATION FOUNDATION (KR) 2021-07-15 US claimed
WO-2021047572-A1 GSK-3β/CHE DOUBLE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 中国药科大学 2021-03-18 WO claimed
CN-112110908-A 1, 3-disubstituted indazole compound and preparation method and application thereof 山东大学 2020-12-22 CN claimed
CN-105218397-B Method for synthesizing 2-azidomethyl-4-nitrobenzoyl chloride 济南大学 2017-05-10 CN claimed
CN-103626705-B 1 (3 benzamido benzyl) 1H indazole 3 Carbox amide and preparation method thereof and anti-viral uses 中国科学院上海药物研究所 2016-12-21 CN claimed
CN-105017569-A Degradable composite tourist commodity packaging film and preparation method thereof JILIN TECHNOLOGY COLLEGE OF ELECTRONIC INFORMATION 2015-11-04 CN claimed
CN-102219800-B Organic substituted boric acid ester, boron affinity functional material using organic substituted boric acid ester as functional monomer as well as preparation and application of organic substituted boric acid ester NANJING UNIVERSITY OF TECHNOLOGY 2015-02-25 CN claimed
CN-104370936-A Novel pyruvate kinase M2 activator and its synthetic method SUZHOU VIVOTIDE BIOTECHNOLOGIES CO LTD 2015-02-25 CN claimed
CN-102219800-A Organic substituted boric acid ester, boron affinity functional material using organic substituted boric acid ester as functional monomer as well as preparation and application of organic substituted boric acid ester NANJING UNIVERSITY OF TECHNOLOGY 2011-10-19 CN claimed
US-7777069-B2 Prodrugs of carbamate inhibitors of IMPDH VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-08-17 US claimed
US-20090093639-A1 Prodrugs of carbamate inhibitors of IMPDH VERTEX PHARMACEUTICAL INCORPORATED (US) 2009-04-09 US claimed
EP-1754705-A2 Antagonists for treatment of CD11/CD18 adhesion receptor mediated disorders Genentech, Inc. (US) 2007-02-21 EP claimed
US-4257915-A USE IN PHOTOPOLYMERIZATION OF ETHYLENICALLY UNSATURATED MONOMERS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1981-03-24 US claimed