SCHEMBL18964376

SCHEMBL18964376

C=CC(=O)N1CCN(c2ncnc3c(/C=C/C)c(-c4c(F)cccc4OC)c(Cl)cc23)CC1

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KRAS P01116 20/20 0.63
EGFR P00533 1/20 0.63
HMOX2 P30519 1/20 0.63
CRYZ Q08257 1/20 0.63
VAT1 Q99536 1/20 0.63
RTN4 Q9NQC3 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16636979 0.90 KRAS (0.78) KRASEGFRHMOX2CRYZVAT1
SCHEMBL21415542 0.87 KRAS (0.64) KRASEGFRHMOX2CRYZVAT1
SCHEMBL29765671 0.82 KRAS (0.69) KRASEGFRHMOX2CRYZVAT1
SCHEMBL16646900 0.82 KRAS (0.69) KRASEGFRHMOX2CRYZVAT1
SCHEMBL16647011 0.81 KRAS (0.63) KRASEGFRHMOX2CRYZVAT1
SCHEMBL29765643 0.81 KRAS (0.63) KRASEGFRHMOX2CRYZVAT1
SCHEMBL29765758 0.81 KRAS (0.80) KRASEGFRHMOX2CRYZVAT1
SCHEMBL16646906 0.81 KRAS (0.80) KRASEGFRHMOX2CRYZVAT1
SCHEMBL19681380 0.80 KRAS (0.63) KRASEGFRHMOX2CRYZVAT1
SCHEMBL18128605 0.79 KRAS (0.75) KRASEGFRHMOX2CRYZVAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017100546-A1 METHODS FOR PREPARATION OF QUINAZOLINE DERIVATIVES ARAXES PHARMA LLC (US) 2017-06-15 WO disclosed