SCHEMBL18965751

SCHEMBL18965751

Cc1ccc2cc3cc(N)sc3cc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.48
CYP1A2 P05177 3/20 0.48
BACE1 P56817 2/20 0.47
TDP1 Q9NUW8 4/20 0.42
MAPT P10636 3/20 0.41
RAB9A P51151 2/20 0.41
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 2/20 0.39
GAA P10253 2/20 0.39
HSD17B10 Q99714 2/20 0.39
NCK1 P16333 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12323 0.84 BACE1 (0.58) CYP2A6CYP1A2BACE1TDP1MAPT
SCHEMBL16471396 0.84 MAPT (0.50) CYP2A6CYP1A2BACE1TDP1MAPT
SCHEMBL17795981 0.81 CYP2A6 (0.52) CYP2A6CYP1A2BACE1TDP1MAPT
SCHEMBL18407859 0.79 BACE1 (0.43) BACE1ALDH1A1TP53SMN1; SMN2CYP3A4
SCHEMBL17934649 0.78 BACE1 (0.50) CYP2A6BACE1TDP1MAPTRAB9A
SCHEMBL4428302 0.77 BACE1 (0.50) CYP2A6BACE1ALDH1A1TP53SMN1; SMN2
SCHEMBL4424142 0.75 BACE1 (0.48) BACE1
SCHEMBL6056946 0.74 CYP1A2 (0.87) CYP2A6CYP1A2BACE1TDP1MAPT
SCHEMBL2463834 0.74 CYP1A2 (0.87) CYP2A6CYP1A2BACE1TDP1MAPT
SCHEMBL4368477 0.74 CYP1A2 (0.87) CYP2A6CYP1A2BACE1TDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3551635-B1 THIENO-INDENO-MONOMERS AND POLYMERS BASF SE (DE) 2021-04-28 EP disclosed
EP-3166949-B1 THIENOTHIOPHENE-ISOINDIGO CLAP CO LTD (KR) 2021-02-17 EP disclosed
WO-2020078815-A1 INDACENO DERIVATIVES AS ORGANIC SEMICONDUCTORS BASF SE (DE) 2020-04-23 WO disclosed
EP-3386989-B1 NAPHTHOINDACENODITHIOPHENES AND POLYMERS BASF SE (DE) 2019-10-23 EP disclosed
WO-2018104367-A2 THIENO-INDENO-MONOMERS AND POLYMERS BASF SE (DE) 2018-06-14 WO disclosed
WO-2017097924-A1 NAPHTHOINDACENODITHIOPHENES AND POLYMERS BASF SE (DE) 2017-06-15 WO disclosed