SCHEMBL1897377

SCHEMBL1897377

CCn1c(C2(O)CCCCO2)nc2c(N3CCOCC3C)nc(Cl)nc21

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTOR P42345 16/20 0.39
PIK3CA P42336 5/20 0.34
PIK3CD O00329 4/20 0.34
PDE4D Q08499 1/20 0.32
ATR Q13535 2/20 0.31
ATRIP Q8WXE1 1/20 0.31
CHEK1 O14757 1/20 0.31
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1896175 0.88 MTOR (0.41) MTORPIK3CAPIK3CDPDE4DATR
SCHEMBL1611450 0.85 MTOR (0.41) MTORPIK3CAPIK3CDPDE4DATR
SCHEMBL1611447 0.85 MTOR (0.41) MTORPIK3CAPIK3CDPDE4DATR
SCHEMBL1612056 0.84 MTOR (0.42) MTORPIK3CAPIK3CDPDE4DATR
SCHEMBL1612053 0.84 MTOR (0.42) MTORPIK3CAPIK3CDPDE4DATR
SCHEMBL1612539 0.81 MTOR (0.41) MTORPIK3CAPIK3CDPDE4DATR
SCHEMBL1612540 0.81 MTOR (0.41) MTORPIK3CAPIK3CDPDE4DATR
SCHEMBL1612580 0.80 MTOR (0.42) MTORPIK3CAPIK3CDPDE4DATR
SCHEMBL1612578 0.80 MTOR (0.42) MTORPIK3CAPIK3CDPDE4DATR
SCHEMBL25279339 0.78 MTOR (0.45) MTORPIK3CAPIK3CDPDE4DATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2498780-A2 N-9-SUBSTITUTED PURINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE F. Hoffmann-La Roche AG (CH) 2012-09-19 EP disclosed
WO-2011058027-A2 N-9-SUBSTITUTED PURINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2011-05-19 WO disclosed