SCHEMBL1897422

SCHEMBL1897422

CCCN1CCC(Oc2cc[c]cc2)CC1

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.68
CARM1 Q86X55 1/20 0.51
PRMT6 Q96LA8 1/20 0.51
DRD2 P14416 5/20 0.47
SLC5A7 Q9GZV3 1/20 0.43
PARP1 P09874 2/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1891613 0.91 HRH3 (0.57) HRH3CARM1PRMT6PARP1MAOA
SCHEMBL5657345 0.87 HRH3 (0.68) HRH3CARM1PRMT6DRD2
SCHEMBL1896242 0.84 HRH3 (0.49) HRH3CARM1PRMT6DRD2PARP1
SCHEMBL20328148 0.84 CARM1 (0.70) HRH3CARM1PRMT6DRD2SLC5A7
SCHEMBL20217556 0.83 HRH3 (0.69) HRH3CARM1PRMT6DRD2PARP1
SCHEMBL1899977 0.82 HRH3 (0.47) HRH3CARM1PRMT6
SCHEMBL188648 0.82 HRH3 (0.63) HRH3CARM1PRMT6MAOAMAOB
SCHEMBL5206619 0.81 HRH3 (1.00) HRH3MAOAMAOB
SCHEMBL19207211 0.78 HRH3 (0.52) HRH3CARM1PRMT6DRD2
SCHEMBL189065 0.77 HRH3 (0.53) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493571-A1 ALKYNYL DERIVATIVES USEFUL AS DPP-1 INHIBITORS Janssen Pharmaceutica, N.V. (BE) 2012-09-05 EP disclosed
WO-2011059731-A1 ALKYNYL DERIVATIVES USEFUL AS DPP-1 INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2011-05-19 WO disclosed