SCHEMBL19001216

SCHEMBL19001216

O=S(=O)(Nc1nccs1)c1cc(Cl)c(NCCCCNC[C@@H]2CCCCCN2)cc1F

nearest known ligand 0.94

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 12/20 0.94
SCN1A P35498 1/20 0.94
CYP3A4 P08684 11/20 0.79
SCN5A Q14524 10/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18992625 0.99 SCN9A (0.95) SCN9ASCN1ACYP3A4SCN5A
SCHEMBL18992589 0.99 SCN9A (0.95) SCN9ASCN1ACYP3A4SCN5A
SCHEMBL20586567 0.99 SCN9A (0.95) SCN9ASCN1ACYP3A4SCN5A
SCHEMBL20167681 0.98 SCN9A (0.94) SCN9ASCN1ACYP3A4SCN5A
SCHEMBL30626708 0.98 SCN9A (0.94) SCN9ASCN1ACYP3A4SCN5A
SCHEMBL18992227 0.97 SCN9A (1.00) SCN9ASCN1ACYP3A4SCN5A
SCHEMBL18992917 0.97 SCN9A (1.00) SCN9ASCN1ACYP3A4SCN5A
SCHEMBL18992225 0.97 SCN9A (1.00) SCN9ASCN1ACYP3A4SCN5A
SCHEMBL18992770 0.93 SCN9A (0.89) SCN9ASCN1ACYP3A4SCN5A
SCHEMBL18992390 0.93 SCN9A (0.89) SCN9ASCN1ACYP3A4SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017106409-A1 DIAMINO-ALKYLAMINO-LINKED ARYLSULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS MERCK SHARP & DOHME CORP. (US) 2017-06-22 WO disclosed