SCHEMBL19001905

SCHEMBL19001905

Brc1cccc2c1-c1ccccc1C21c2ccccc2-c2c(-c3cccc(-c4ccccc4)c3)cccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 6/20 0.44
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
PTGER1 P34995 1/20 0.34
PTGER4 P35408 1/20 0.34
PTGER3 P43115 1/20 0.34
PTGER2 P43116 1/20 0.34
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
KMO O15229 1/20 0.31
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31
MAOA P21397 1/20 0.31
MEN1 O00255 1/20 0.30
APAF1 O14727 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23222599 0.91 PDK2 (0.46) PDK2ALDH1A1MAPK1CRHBPCRHR2
SCHEMBL19001863 0.91 PDK2 (0.49) PDK2ALDH1A1MAPK1CA1CA2
SCHEMBL30257749 0.89 PDK2 (0.41) PDK2PTGER1PTGER4PTGER3PTGER2
SCHEMBL25222229 0.89 PDK2 (0.41) PDK2PTGER1PTGER4PTGER3PTGER2
SCHEMBL19001698 0.88 PDK2 (0.42) PDK2ALDH1A1MAPK1PTGER1PTGER4
SCHEMBL19001985 0.87 PDK2 (0.43) PDK2ALDH1A1MAPK1MEN1APAF1
SCHEMBL15840175 0.87 PDK2 (0.46) PDK2ALDH1A1MAPK1MEN1APAF1
SCHEMBL15840172 0.87 PDK2 (0.46) PDK2ALDH1A1MAPK1MEN1APAF1
SCHEMBL19001861 0.87 PDK2 (0.43) PDK2ALDH1A1MAPK1CRHBPCRHR2
SCHEMBL19001702 0.87 PDK2 (0.46) PDK2ALDH1A1MAPK1MEN1APAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3390365-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2021-04-14 EP disclosed
WO-2017102063-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2017-06-22 WO disclosed