SCHEMBL19002865

SCHEMBL19002865

CCC(C)N1CCN(c2ccccc2)CC1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.44
DRD2 P14416 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
GFER P55789 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
DPP4 P27487 2/20 0.39
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
NOTUM Q6P988 1/20 0.36
CHRM4 P08173 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17897247 0.84 KDM4E (0.41) CHRNA7DRD2SIGMAR1KDM4EALDH1A1
SCHEMBL17897242 0.84 KDM4E (0.41) CHRNA7DRD2SIGMAR1KDM4EALDH1A1
SCHEMBL19003675 0.84 KDM4E (0.41) CHRNA7DRD2SIGMAR1KDM4EALDH1A1
SCHEMBL10269322 0.74 CHRNA7 (0.56) CHRNA7DRD2SIGMAR1KDM4EALDH1A1
SCHEMBL12662987 0.72 ESR1 (0.52) CHRNA7DRD2SIGMAR1ADRA2AADRA2B
SCHEMBL13380548 0.72 ESR1 (0.52) CHRNA7DRD2SIGMAR1ADRA2AADRA2B
SCHEMBL3567530 0.72 ESR1 (0.52) CHRNA7DRD2SIGMAR1ADRA2AADRA2B
SCHEMBL10438606 0.72 KDM4E (0.43) CHRNA7DRD2SIGMAR1KDM4EALDH1A1
SCHEMBL10438605 0.72 KDM4E (0.43) CHRNA7DRD2SIGMAR1KDM4EALDH1A1
SCHEMBL28851967 0.71 CHRNA7 (0.49) CHRNA7DRD2SIGMAR1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2938344-B1 PIPERAZINE-SUBSTITUTED [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINE COMPOUNDS WITH A2A ANTAGONIST PROPERTIES MERCK SHARP & DOHME (US) 2017-06-21 EP disclosed