SCHEMBL19005817

SCHEMBL19005817

CC(C)(C)OC(=O)N1CCc2c(C(C)(C)O)n[nH]c2C1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.44
ESR2 Q92731 1/20 0.41
NR1H2 P55055 2/20 0.41
PARP1 P09874 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
MAPK1 P28482 1/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
USP2 O75604 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
F12 P00748 2/20 0.36
MKNK1 Q9BUB5 2/20 0.36
DPP4 P27487 1/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
RBP4 P02753 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21237549 0.92 ADORA1 (0.45) ADORA1ESR2NR1H2PARP1TNKS2
SCHEMBL17868704 0.90 ESR2 (0.41) ADORA1ESR2NR1H2PARP1TNKS2
SCHEMBL1424003 0.89 DPP4 (0.46) ADORA1ESR2NR1H2PARP1TNKS2
SCHEMBL17229883 0.84 ADORA1 (0.45) ADORA1ESR2NR1H2PARP1TNKS2
SCHEMBL17317597 0.83 ADORA1 (0.44) ADORA1ESR2NR1H2PARP1TNKS2
SCHEMBL17317969 0.83 ADORA1 (0.50) ADORA1ESR2NR1H2PARP1TNKS2
SCHEMBL19643783 0.83 ADORA1 (0.44) ADORA1ESR2NR1H2PARP1TNKS2
SCHEMBL17223055 0.82 ADORA1 (0.49) ADORA1ESR2NR1H2PARP1TNKS2
SCHEMBL10296218 0.82 ESR2 (0.43) ADORA1ESR2NR1H2PARP1TNKS2
SCHEMBL21994486 0.81 ADORA1 (0.43) ADORA1ESR2NR1H2PARP1TNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107207504-B Phthalazinone derivatives, preparation method and use thereof 四川科伦博泰生物医药股份有限公司 2020-03-10 CN disclosed
WO-2017101796-A1 PHTHALAZINONE DERIVATIVE, AND PREPARATION METHOD AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-22 WO disclosed