SCHEMBL19033604

SCHEMBL19033604

BC(B)(B)Oc1cnc(C(=O)Nc2cc(F)c(F)c([C@]3(C)CS(=O)(=O)N(C)C(=N)N3)c2)cn1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.56
BACE2 Q9Y5Z0 5/20 0.56
CTSD P07339 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19033573 0.93 BACE1 (0.49) BACE1BACE2
SCHEMBL15892964 0.93 BACE1 (0.56) BACE1BACE2CTSD
SCHEMBL19033660 0.92 BACE1 (0.49) BACE1BACE2CTSD
SCHEMBL10328853 0.90 BACE1 (0.68) BACE1BACE2CTSD
SCHEMBL19033661 0.90 BACE1 (0.49) BACE1BACE2CTSD
SCHEMBL10328868 0.89 BACE1 (0.57) BACE1BACE2
SCHEMBL10328867 0.88 BACE1 (0.55) BACE1BACE2
SCHEMBL10328891 0.88 BACE1 (0.60) BACE1BACE2CTSD
SCHEMBL10328873 0.87 BACE1 (0.56) BACE1BACE2CTSD
SCHEMBL19033577 0.87 BACE1 (0.47) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9687494-B2 Iminothiadiazine dioxide compounds as BACE inhibitors, compositions, and their use MERCK SHARP & DOHME CORP. (US) 2017-06-27 US disclosed