SCHEMBL1908335

SCHEMBL1908335

CC(=O)Nc1cccc(-c2cnc3oc(-c4ccc(C5(N)CCC5)cc4)c(-c4ccccc4)c3n2)c1.NC1(c2ccc(-c3oc4ncc(-c5cccnc5)nc4c3-c3ccccc3)cc2)CCC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 12/20 0.48
AKT2 P31751 7/20 0.48
CYP2C8 P10632 2/20 0.48
CYP2D6 P10635 2/20 0.48
CYP2C9 P11712 2/20 0.48
AKT3 Q9Y243 2/20 0.48
ATR Q13535 3/20 0.46
GSK3B P49841 1/20 0.46
BRAF P15056 1/20 0.44
NPC1 O15118 1/20 0.44
TP53 P04637 1/20 0.44
STAT1 P42224 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PLK1 P53350 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1902022 0.96 AKT1 (0.49) AKT1AKT2CYP2C8CYP2D6CYP2C9
SCHEMBL1908337 0.88 AKT1 (0.39) AKT1AKT2CYP2C8CYP2D6CYP2C9
SCHEMBL1900959 0.87 AKT1 (0.52) AKT1AKT2CYP2D6CYP2C9AKT3
SCHEMBL1903012 0.82 AKT1 (0.51) AKT1AKT2ATR
SCHEMBL1902768 0.81 NPC1 (0.42) AKT1AKT2CYP2C8CYP2D6CYP2C9
SCHEMBL1905644 0.80 AKT1 (0.51) AKT1AKT2
SCHEMBL1904321 0.79 AKT1 (0.47) AKT1AKT2
SCHEMBL1900984 0.78 AKT1 (0.40) AKT1AKT2ATRGSK3B
SCHEMBL1907297 0.77 AKT1 (0.53) AKT1AKT2
SCHEMBL1903876 0.75 AKT1 (0.50) AKT1AKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496566-A1 AKT / PKB INHIBITORS Almac Discovery Limited (GB) 2012-09-12 EP claimed
WO-2011055115-A1 AKT / PKB INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2011-05-12 WO claimed