SCHEMBL19086229

SCHEMBL19086229

CC1(C)CC(=O)c2c(C(F)F)nn(-c3ccc(C(N)=O)c(NC4CCC(NCC(=O)O)CC4)c3)c2C1

nearest known ligand 0.81

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 20/20 0.81
HSP90AA1 P07900 19/20 0.81
HSP90B1 P14625 6/20 0.63
TRAP1 Q12931 6/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1219609 0.90 HSP90AA1 (1.00) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL1219606 0.90 HSP90AA1 (1.00) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL16161869 0.89 HSP90AB1 (0.80) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL1220841 0.88 HSP90AA1 (0.85) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL1220380 0.88 HSP90AA1 (0.85) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL16161783 0.88 HSP90AA1 (0.81) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL38654958 0.88 HSP90AA1 (0.81) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL1219082 0.88 HSP90AA1 (1.00) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL8122876 0.87 HSP90AA1 (0.82) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL1220579 0.87 HSP90AA1 (0.80) HSP90AB1HSP90AA1HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2380879-B1 Tetrahydroindolone and tetrahydroindazolone derivatives ESANEX INC (US) 2017-07-12 EP claimed