SCHEMBL19086376

SCHEMBL19086376

CN(C(=O)O)C1(CN2CCC(CNC(=O)c3cc(C(F)(F)F)cc(C(F)(F)F)c3)CC2)CCCC1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 11/20 0.60
CACNA1I Q9P0X4 11/20 0.60
MCHR1 Q99705 3/20 0.45
HTR1A P08908 1/20 0.45
ADRA2A P08913 1/20 0.45
ADRA1A P35348 1/20 0.45
HTR2B P41595 1/20 0.45
CCR2 P41597 1/20 0.41
CACNA1G O43497 1/20 0.40
CACNA1H O95180 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14769919 0.85 KCNH2 (0.66) KCNH2CACNA1IMCHR1HTR1AADRA2A
SCHEMBL19112594 0.83 KCNH2 (0.63) KCNH2CACNA1IMCHR1HTR1AADRA2A
SCHEMBL1427896 0.83 KCNH2 (0.62) KCNH2CACNA1IMCHR1HTR1AADRA2A
SCHEMBL4278940 0.83 KCNH2 (0.60) KCNH2CACNA1IMCHR1HTR1AADRA2A
SCHEMBL19112701 0.81 KCNH2 (0.60) KCNH2CACNA1IMCHR1HTR1AADRA2A
SCHEMBL7797275 0.80 CACNA1I (0.60) KCNH2CACNA1IMCHR1HTR1AADRA2A
SCHEMBL1428777 0.80 KCNH2 (0.57) KCNH2CACNA1IMCHR1HTR1AADRA2A
SCHEMBL4270480 0.80 KCNH2 (0.55) KCNH2CACNA1IMCHR1HTR1AADRA2A
SCHEMBL1428180 0.80 KCNH2 (0.59) KCNH2CACNA1IMCHR1HTR1AADRA2A
SCHEMBL4278118 0.80 KCNH2 (0.59) KCNH2CACNA1IMCHR1HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3189839-A1 N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS Taro Pharmaceuticals Inc. (CA) 2017-07-12 EP disclosed