SCHEMBL19089053

SCHEMBL19089053

Cc1nc2c(F)cc(-c3nc(Nc4ccc5c(n4)CCN(CCNO)C5)ncc3F)cc2n1C(C)(C)C

nearest known ligand 0.88

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.88
CDK2 P24941 20/20 0.88
CDK6 Q00534 20/20 0.88
CDK1 P06493 7/20 0.88
CDK7 P50613 7/20 0.88
CDK9 P50750 7/20 0.88
CDK5 Q00535 7/20 0.88
CCNA2 P20248 1/20 0.82
CCND3 P30281 1/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19089046 0.94 CDK4 (1.00) CDK4CDK2CDK6CDK1CDK7
SCHEMBL19089189 0.93 CDK4 (0.88) CDK4CDK2CDK6CDK1CDK7
SCHEMBL19089056 0.92 CDK4 (1.00) CDK4CDK2CDK6CDK1CDK7
SCHEMBL19089208 0.91 CDK4 (1.00) CDK4CDK2CDK6CDK1CDK7
SCHEMBL22010578 0.91 CDK4 (0.92) CDK4CDK2CDK6CDK1CDK7
SCHEMBL19089188 0.91 CDK4 (0.88) CDK4CDK2CDK6CDK1CDK7
SCHEMBL19089084 0.91 CDK4 (0.88) CDK4CDK2CDK6CDK1CDK7
SCHEMBL22010371 0.90 CDK4 (0.86) CDK4CDK2CDK6CDK1CDK7
SCHEMBL22261811 0.90 CDK4 (0.87) CDK4CDK2CDK6CDK1CDK7
SCHEMBL22010370 0.90 CDK4 (0.89) CDK4CDK2CDK6CDK1CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114512-A1 NITROGEN-CONTAINING FUSED HETEROCYCLIC COMPOUND, AS WELL AS PREPARATION METHOD, INTERMEDIATE, COMPOSITION AND APPLICATION THEREOF 上海医药集团股份有限公司 2017-07-06 WO disclosed