SCHEMBL19101136

SCHEMBL19101136

N#Cc1cccc(NC(=O)c2nc(-c3ccccc3)cnc2N)c1

nearest known ligand 0.88

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ATR Q13535 20/20 0.88
PRKDC P78527 7/20 0.88
ATM Q13315 2/20 0.64
CYP3A4 P08684 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2487055 0.94 ATR (1.00) ATRPRKDCATMCYP3A4
SCHEMBL2483560 0.91 ATR (1.00) ATRPRKDCCYP3A4
SCHEMBL2485447 0.88 ATR (1.00) ATRPRKDCATM
SCHEMBL30667685 0.85 ATR (1.00) ATRPRKDCATMCYP3A4
SCHEMBL2480842 0.85 ATR (1.00) ATRPRKDCATMCYP3A4
SCHEMBL19101062 0.83 ATR (0.87) ATRPRKDCATMCYP3A4
SCHEMBL3459870 0.81 ATR (0.74) ATRPRKDC
SCHEMBL2486940 0.80 ATR (1.00) ATRPRKDCATMCYP3A4
Hydrochloric Acid SCHEMBL3159476 0.80 GSK3B (0.75) ATRPRKDC
SCHEMBL3462673 0.80 ATR (0.66) ATRPRKDCATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9701674-B2 Substituted pyrazines as ATR kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2017-07-11 US disclosed