SCHEMBL19102407

SCHEMBL19102407

CC[C@H]1CC[C@@H](N(C)Cc2ccccc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.52
HRH4 Q9H3N8 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49
SLC18A3 Q16572 1/20 0.47
ALDH1A1 P00352 2/20 0.44
TSHR P16473 1/20 0.44
DDB1 Q16531 1/20 0.43
CRBN Q96SW2 1/20 0.43
OPRM1 P35372 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
KDM4E B2RXH2 2/20 0.42
NAAA Q02083 1/20 0.42
AOC3 Q16853 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19390970 1.00 GRIN2B (0.52) GRIN2BHRH4HRH3SLC18A3ALDH1A1
SCHEMBL3375289 0.89 GRIN2B (0.61) GRIN2BHRH4HRH3SLC18A3ALDH1A1
SCHEMBL32688193 0.84 SLC6A2 (0.49) GRIN2BSLC18A3ALDH1A1TSHRKDM4E
SCHEMBL11251947 0.83 HRH3 (0.67) GRIN2BHRH4HRH3SLC18A3ALDH1A1
SCHEMBL13744978 0.82 GRIN2B (0.55) GRIN2BHRH4HRH3SLC18A3ALDH1A1
SCHEMBL14506713 0.82 GRIN2B (0.55) GRIN2BHRH4HRH3SLC18A3ALDH1A1
SCHEMBL12680890 0.82 GRIN2B (0.55) GRIN2BHRH4HRH3SLC18A3ALDH1A1
Bromide SCHEMBL11253051 0.82 HRH3 (0.65) GRIN2BHRH4HRH3SLC18A3ALDH1A1
SCHEMBL531089 0.82 HRH3 (0.70) GRIN2BHRH4HRH3SLC18A3ALDH1A1
SCHEMBL16367134 0.81 GRIN2B (0.54) GRIN2BHRH4HRH3SLC18A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9701666-B2 1,4-pyridone bicyclic heteroaryl compounds Epizyme, Inc. (US) 2017-07-11 US disclosed