SCHEMBL19112833

SCHEMBL19112833

CC(C)(C)C1CCN(CC(=O)N2CCC(CNC(=P)c3cc(F)cc(C(F)(F)F)c3)CC2)CC1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.48
CACNA1I Q9P0X4 8/20 0.48
CACNA1G O43497 1/20 0.47
CACNA1H O95180 1/20 0.47
CCR2 P41597 1/20 0.38
TACR1 P25103 1/20 0.38
RORC P51449 1/20 0.37
CXCR3 P49682 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4276605 0.92 KCNH2 (0.58) KCNH2CACNA1ICACNA1GCACNA1HRORC
SCHEMBL13569753 0.90 KCNH2 (0.47) KCNH2CACNA1ICACNA1GCACNA1HCCR2
SCHEMBL4275245 0.86 KCNH2 (0.65) KCNH2CACNA1ICACNA1GCACNA1HRORC
SCHEMBL4272256 0.86 KCNH2 (0.65) KCNH2CACNA1ICACNA1GCACNA1HRORC
SCHEMBL19112606 0.84 CACNA1I (0.42) KCNH2CACNA1ICACNA1GCACNA1HCCR2
SCHEMBL4274763 0.82 KCNH2 (0.57) KCNH2CACNA1ICACNA1GCACNA1HCCR2
SCHEMBL4271076 0.82 KCNH2 (0.55) KCNH2CACNA1ICACNA1GCACNA1HCCR2
SCHEMBL19113096 0.82 KCNH2 (0.60) KCNH2CACNA1ICACNA1GCACNA1HCCR2
SCHEMBL4277349 0.81 KCNH2 (0.56) KCNH2CACNA1ICACNA1GCACNA1HCCR2
SCHEMBL4275313 0.81 KCNH2 (0.56) KCNH2CACNA1ICACNA1GCACNA1HCCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3189839-A1 N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS Taro Pharmaceuticals Inc. (CA) 2017-07-12 EP disclosed