SCHEMBL19182802

SCHEMBL19182802

C[C@H](C(=O)N[C@H]1Cc2ccccc2[C@H]1O)c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 9/20 0.62
PSEN1 P49768 1/20 0.44
PSEN2 P49810 1/20 0.44
APH1B Q8WW43 1/20 0.44
NCSTN Q92542 1/20 0.44
APH1A Q96BI3 1/20 0.44
PSENEN Q9NZ42 1/20 0.44
CNR1 P21554 1/20 0.44
PYGL P06737 2/20 0.42
SOAT1 P35610 1/20 0.42
MAPK14 Q16539 1/20 0.42
KCNQ2 O43526 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19200149 1.00 GRM7 (0.62) GRM7PSEN1PSEN2APH1BNCSTN
SCHEMBL19182810 1.00 GRM7 (0.62) GRM7PSEN1PSEN2APH1BNCSTN
SCHEMBL19183401 1.00 GRM7 (0.62) GRM7PSEN1PSEN2APH1BNCSTN
SCHEMBL19182811 1.00 GRM7 (0.62) GRM7PSEN1PSEN2APH1BNCSTN
SCHEMBL19200896 1.00 GRM7 (0.62) GRM7PSEN1PSEN2APH1BNCSTN
SCHEMBL20678754 1.00 GRM7 (0.62) GRM7PSEN1PSEN2APH1BNCSTN
SCHEMBL20678612 1.00 GRM7 (0.62) GRM7PSEN1PSEN2APH1BNCSTN
SCHEMBL20678603 1.00 GRM7 (0.62) GRM7PSEN1PSEN2APH1BNCSTN
SCHEMBL20678605 1.00 GRM7 (0.62) GRM7PSEN1PSEN2APH1BNCSTN
SCHEMBL20678619 0.90 GRM7 (0.72) GRM7CNR1PYGLMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190031599-A1 INDANE DERIVATIVES AS MGLUR7 MODULATORS TAKEDA CAMBRIDGE LIMITED (GB) 2019-01-31 US claimed
EP-3408256-A1 INDANE DERIVATIVES AS MGLUR7 MODULATORS Takeda Pharmaceutical Company Limited (JP) 2018-12-05 EP claimed
WO-2017131221-A1 INDANE DERIVATIVES AS MGLUR7 MODULATORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-08-03 WO claimed
US-20190031599-A1 INDANE DERIVATIVES AS MGLUR7 MODULATORS TAKEDA CAMBRIDGE LIMITED (GB) 2019-01-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190031599-A1 INDANE DERIVATIVES AS MGLUR7 MODULATORS GRM7, GRIN2B, GRM1 GRM7 1/4885PSEN1 1092/4885PSEN2 903/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.