SCHEMBL19192542

SCHEMBL19192542

CCN(C)Cc1ccc(C(=O)Nc2ccc(C)c(Nc3nccc(-c4cccnc4)n3)c2)cc1Br

nearest known ligand 0.75

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 15/20 0.75
BCR P11274 11/20 0.75
LYN P07948 2/20 0.75
PDGFRA P16234 8/20 0.70
PDGFRB P09619 4/20 0.70
EGFR P00533 1/20 0.68
PRKCA P17252 1/20 0.68
KIT P10721 3/20 0.67
ABL2 P42684 2/20 0.66
MAPK8 P45983 1/20 0.65
MAPK9 P45984 1/20 0.65
MAPK10 P53779 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3568536 0.94 ABL1 (0.73) ABL1BCRLYNPDGFRAPDGFRB
SCHEMBL3566747 0.94 ABL1 (0.75) ABL1BCRLYNPDGFRAPDGFRB
SCHEMBL28755616 0.88 ABL1 (0.80) ABL1BCRLYNPDGFRAPDGFRB
SCHEMBL3568761 0.88 ABL1 (0.89) ABL1BCRLYNPDGFRAPDGFRB
Diethylamine SCHEMBL3568539 0.87 PDGFRA (0.74) ABL1BCRLYNPDGFRAPDGFRB
Dimethylamine SCHEMBL3566750 0.87 ABL1 (0.79) ABL1BCRLYNPDGFRAPDGFRB
SCHEMBL13157377 0.87 ABL1 (0.81) ABL1BCRLYNPDGFRAPDGFRB
SCHEMBL3563459 0.86 ABL1 (1.00) ABL1BCRLYNPDGFRAPDGFRB
SCHEMBL3562697 0.86 ABL1 (0.89) ABL1BCRLYNPDGFRAPDGFRB
SCHEMBL3561315 0.85 ABL1 (0.88) ABL1BCRLYNPDGFRAPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1702917-B1 AMIDE DERIVATIVE AND MEDICINE NIPPON SHINYAKU CO LTD (JP) 2017-08-02 EP disclosed