SCHEMBL19210478

SCHEMBL19210478

COC(=O)NCc1cnccn1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.50
HDAC3 O15379 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
NAMPT P43490 2/20 0.45
CYP2C9 P11712 1/20 0.45
VNN1 O95497 2/20 0.44
RAB9A P51151 1/20 0.43
CHRM4 P08173 1/20 0.42
POLB P06746 1/20 0.42
SPR P35270 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
IDO1 P14902 1/20 0.40
PIK3CA P42336 1/20 0.40
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30089199 0.84 NAMPT (0.48) HPGDSHDAC3HDAC1HDAC2HDAC6
SCHEMBL1265671 0.84 NAMPT (0.48) HPGDSHDAC3HDAC1HDAC2HDAC6
SCHEMBL29602711 0.82 NPSR1 (0.50) HPGDSHDAC3HDAC1HDAC2HDAC6
SCHEMBL3003567 0.82 NPSR1 (0.50) HPGDSHDAC3HDAC1HDAC2HDAC6
SCHEMBL1933893 0.80 HDAC3 (0.51) HPGDSHDAC3HDAC1HDAC2HDAC6
SCHEMBL9245 0.79 HDAC3 (0.48) HPGDSHDAC3HDAC1HDAC2HDAC6
SCHEMBL23022741 0.79 HDAC3 (0.50) HPGDSHDAC3HDAC1HDAC2HDAC6
SCHEMBL21246171 0.79 RECQL (0.53) HPGDSHDAC3HDAC1HDAC2HDAC6
SCHEMBL3003564 0.79 HDAC3 (0.50) HPGDSHDAC3HDAC1HDAC2HDAC6
SCHEMBL29884167 0.79 RECQL (0.53) HPGDSHDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2699557-B1 3-(OXAZOL-2-YL-ETHOXY)- AND 3-(THIAZOL-2-YL-ETHOXY)-BENZAMIDE DERIVATIVES AS ANTI-BACTERIAL AGENTS BIOTA SCIENT MANAGEMENT (AU) 2017-08-16 EP claimed
WO-2020023793-A1 PEGYLATED PRODRUGS OF PHENOLIC TRPV1 AGONISTS Concentric Analgesics, Inc. (US) 2020-01-30 WO disclosed