Ethyne

Ethyne

SCHEMBL1921187

C#C.O=CNCc1nccs1

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.42
TRPM5 Q9NZQ8 1/20 0.39
FDPS P14324 1/20 0.39
KDM1A O60341 2/20 0.38
MAOB P27338 1/20 0.38
ADH1B P00325 1/20 0.34
ADH1C P00326 1/20 0.34
ADH1A P07327 1/20 0.34
ADH7 P40394 1/20 0.34
SLC6A3 Q01959 3/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
DRD4 P21917 1/20 0.34
PSMD14 O00487 1/20 0.33
STAMBP O95630 1/20 0.33
COPS5 Q92905 1/20 0.33
NTRK1 P04629 1/20 0.32
ALDH1A1 P00352 2/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1258299 0.96
SCHEMBL1998111 0.78 DRD4 (0.41) CYP2C19TRPM5FDPSKDM1AMAOB
SCHEMBL2311217 0.78 CYP2C19 (0.46) CYP2C19TRPM5FDPSKDM1AMAOB
SCHEMBL14216629 0.76 CYP2C19 (0.43) CYP2C19TRPM5FDPSKDM1AMAOB
SCHEMBL2000599 0.75 DRD4 (0.38) CYP2C19TRPM5FDPSADH1BADH1C
SCHEMBL22593333 0.71
SCHEMBL4574553 0.71
SCHEMBL1628173 0.71
SCHEMBL18884390 0.70
SCHEMBL13548386 0.70 CYP2C19 (0.44) CYP2C19TRPM5FDPSKDM1AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981854-B1 ARYLPROPIONAMIDE, ARYLACRYLAMIDE, ARYLPROPYNAMIDE, OR ARYLMETHYLUREA ANALOGS AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-06-01 EP claimed