SCHEMBL19216879

SCHEMBL19216879

Cc1cccc(NC(=O)Nc2ccc(-c3nc(N4CCOCC4)c4cc(CN(C)C)cn4n3)cc2)c1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 10/20 0.59
PIK3R1 P27986 3/20 0.54
MTOR P42345 15/20 0.50
PIK3CG P48736 5/20 0.50
PIK3CD O00329 2/20 0.50
KDR P35968 1/20 0.47
FLT3 P36888 1/20 0.47
PIK3CB P42338 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16611751 0.93 PIK3CA (0.63) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16611594 0.92 PIK3CA (0.59) PIK3CAPIK3R1MTORPIK3CGPIK3CD
SCHEMBL16611516 0.89 PIK3CA (0.57) PIK3CAPIK3R1MTORPIK3CGPIK3CD
SCHEMBL16611293 0.89 PIK3CA (0.65) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16727835 0.89 PIK3CA (0.62) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16611050 0.89 PIK3CA (0.72) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16612099 0.89 PIK3CA (0.62) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16611517 0.88 PIK3CA (0.75) PIK3CAPIK3R1MTORPIK3CG
SCHEMBL16611755 0.87 PIK3CA (0.61) PIK3CAPIK3R1MTOR
SCHEMBL16622894 0.87 PIK3CA (0.60) PIK3CAPIK3R1MTORPIK3CGPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9724352-B2 Pyrrolo[2,1-F[1,2,4]triazine compounds, preparation methods and applications thereof SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2017-08-08 US disclosed