SCHEMBL19217032

SCHEMBL19217032

COC1CCCN(c2nc(-c3cnc(N)cc3C(F)(F)F)nn3cc(CN4CCN(S(C)(=O)=O)CC4)cc23)C1

nearest known ligand 0.76

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 19/20 0.76
PIK3R1 P27986 12/20 0.73
PIK3CD O00329 4/20 0.59
PIK3CB P42338 4/20 0.59
RAF1 P04049 1/20 0.59
PIK3CG P48736 3/20 0.45
MTOR P42345 4/20 0.38
RICTOR Q6R327 2/20 0.36
RPTOR Q8N122 2/20 0.36
MAPKAP1 Q9BPZ7 2/20 0.36
MLST8 Q9BVC4 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19216878 0.86 PIK3CA (0.56) PIK3CAPIK3R1PIK3CDPIK3CBRAF1
SCHEMBL16611564 0.86 PIK3CA (1.00) PIK3CAPIK3R1PIK3CDPIK3CBRAF1
SCHEMBL16611611 0.84 PIK3CA (1.00) PIK3CAPIK3R1PIK3CDPIK3CBRAF1
SCHEMBL16611392 0.80 PIK3CA (1.00) PIK3CAPIK3R1PIK3CDPIK3CBRAF1
SCHEMBL16611391 0.80 PIK3CA (1.00) PIK3CAPIK3R1PIK3CDPIK3CBRAF1
SCHEMBL19216996 0.79 PIK3CA (0.75) PIK3CAPIK3R1PIK3CDPIK3CBRAF1
SCHEMBL16727841 0.76 PIK3CA (0.82) PIK3CAPIK3R1PIK3CDPIK3CBRAF1
SCHEMBL16727840 0.74 PIK3CA (0.81) PIK3CAPIK3R1PIK3CDPIK3CBRAF1
Risovalisib SCHEMBL16622890 0.74 PIK3CA (1.00) PIK3CAPIK3R1PIK3CDPIK3CBRAF1
SCHEMBL16713180 0.73 PIK3CA (0.76) PIK3CAPIK3R1PIK3CDPIK3CBRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9724352-B2 Pyrrolo[2,1-F[1,2,4]triazine compounds, preparation methods and applications thereof SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2017-08-08 US disclosed