SCHEMBL19217765

SCHEMBL19217765

COc1ccc(Nc2ncc(F)c(N[C@H]3[C@@H](C(N)=O)[C@@H]4C=C[C@H]3C4)n2)cc1C

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 10/20 0.71
KDR P35968 9/20 0.71
AURKB Q96GD4 8/20 0.71
ALK Q9UM73 3/20 0.71
AURKA O14965 2/20 0.71
LCK P06239 2/20 0.71
PDGFRA P16234 2/20 0.71
FLT3 P36888 2/20 0.71
SYK P43405 2/20 0.71
INSR P06213 2/20 0.71
MET P08581 2/20 0.71
CDC7 O00311 1/20 0.71
PLK4 O00444 1/20 0.71
CHEK1 O14757 1/20 0.71
DCLK1 O15075 1/20 0.71
PDPK1 O15530 1/20 0.71
DAPK3 O43293 1/20 0.71
JAK2 O60674 1/20 0.71
ROCK2 O75116 1/20 0.71
PRKD3 O94806 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12952297 0.89 IRAK4 (0.74) IRAK4KDRAURKBALKAURKA
SCHEMBL1001618 0.89 IRAK4 (0.74) IRAK4KDRAURKBALKAURKA
Hydrochloric Acid SCHEMBL1988148 0.88 IRAK4 (0.73) IRAK4KDRAURKBALKAURKA
SCHEMBL1002524 0.87 KDR (0.68) IRAK4KDRAURKBALKAURKA
SCHEMBL3553074 0.87 KDR (0.68) IRAK4KDRAURKBALKAURKA
SCHEMBL1002521 0.87 KDR (0.68) IRAK4KDRAURKBALKAURKA
SCHEMBL1003397 0.87 KDR (0.61) IRAK4KDRAURKBALKAURKA
SCHEMBL1000684 0.87 KDR (0.74) IRAK4KDRAURKBALKAURKA
SCHEMBL1000681 0.87 KDR (0.74) IRAK4KDRAURKBALKAURKA
SCHEMBL1000682 0.87 KDR (0.74) IRAK4KDRAURKBALKAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9725419-B2 Cycloalkyl substituted pyrimidinediamine compounds and their uses RIGEL PHARMACEUTICALS, INC. (US) 2017-08-08 US disclosed