SCHEMBL1923014

SCHEMBL1923014

CC(=O)C(C)Cc1ccc(Cl)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
CYP3A4 P08684 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP2D6 P10635 1/20 0.49
ALOX15 P16050 1/20 0.49
EPHX1 P07099 1/20 0.49
HDAC8 Q9BY41 5/20 0.48
CYP2C9 P11712 2/20 0.48
P2RX7 Q99572 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
IDO1 P14902 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
MC4R P32245 2/20 0.44
MAPK1 P28482 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21400207 1.00 GAA (0.51) GAACYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL14198757 1.00 GAA (0.51) GAACYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL6005671 0.86 CYP3A4 (0.52) GAACYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL9780834 0.86 CYP3A4 (0.52) GAACYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL14198754 0.81 HDAC8 (0.57) EPHX1HDAC8HDAC3HDAC1HDAC2
SCHEMBL28322156 0.81 HDAC8 (0.47) GAACYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL15745971 0.81 HDAC8 (0.57) EPHX1HDAC8HDAC3HDAC1HDAC2
SCHEMBL6306721 0.81 CYP3A4 (0.47) GAACYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL26431186 0.79 GAA (0.48) GAACYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL21400206 0.79 NPC1 (0.46) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2328902-A1 PYRAZOLO [5,1-B]OXAZOLE DERIVATIVES AS CRF1 ANTAGONISTS Novartis AG (CH) 2011-06-08 EP disclosed
WO-2010015628-A1 PYRAZOLO [5,1-B] OXAZOLE DERIVATIVES AS CRF1 ANTAGONISTS NOVARTIS AG (CH) 2010-02-11 WO disclosed