SCHEMBL19230837

SCHEMBL19230837

OC(O)c1ccc2c(c1)CCC(c1ccc(OCc3c(-c4c(Cl)cccc4Cl)noc3C3CC3)cc1C(F)(F)F)O2

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.52
FABP1 P07148 2/20 0.47
FXR2 P51116 1/20 0.47
HSD17B13 Q7Z5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230559 0.88 NR1H4 (0.69) NR1H4FXR2HSD17B13
SCHEMBL19230778 0.88 NR1H4 (0.59) NR1H4FXR2HSD17B13
SCHEMBL19231004 0.84 NR1H4 (0.54) NR1H4
SCHEMBL19230542 0.80 NR1H4 (0.58) NR1H4FABP1FXR2
SCHEMBL20661679 0.80 NR1H4 (0.76) NR1H4FABP1
SCHEMBL19230515 0.79 NR1H4 (0.74) NR1H4FXR2HSD17B13
SCHEMBL19230625 0.79 NR1H4 (0.74) NR1H4FXR2HSD17B13
SCHEMBL19230541 0.79 NR1H4 (0.74) NR1H4FXR2HSD17B13
SCHEMBL19230836 0.79 NR1H4 (0.56) NR1H4FXR2HSD17B13
SCHEMBL19230557 0.79 NR1H4 (0.71) NR1H4FXR2HSD17B13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed