SCHEMBL19233286

SCHEMBL19233286

C=C(N)Nc1c(F)ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)c1F

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.56
BRAF P15056 10/20 0.55
NPC1 O15118 1/20 0.46
POLB P06746 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CYP2C9 P11712 1/20 0.46
RAF1 P04049 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19233576 0.86 BRAF (0.59) KDRBRAFNPC1POLBHTT
SCHEMBL20577750 0.83 KDR (0.50) KDRBRAFCYP2C9
SCHEMBL20577950 0.81 PTGS1 (0.56) KDRBRAFCYP2C9
SCHEMBL20577764 0.80 KDR (0.54) KDRBRAFCYP2C9RAF1
SCHEMBL26075765 0.78 BRAF (0.54) BRAFCYP2C9RAF1
SCHEMBL1698051 0.78 KDR (0.53) KDRBRAFCYP2C9RAF1
SCHEMBL26075623 0.77 BRAF (0.57) KDRBRAFCYP2C9
SCHEMBL26075773 0.76 BRAF (0.53) KDRBRAFCYP2C9
SCHEMBL5004766 0.75 BRAF (0.59) BRAFCYP2C9
SCHEMBL2856788 0.74 BRAF (0.51) KDRBRAFCYP2C9RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017135589-A9 PYRIDINE DERIVATIVE INHIBITING RAF KINASE AND VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR, METHOD FOR PREPARING SAME, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND USE THEREOF 삼진제약주식회사 2017-10-19 WO disclosed
WO-2017135589-A1 PYRIDINE DERIVATIVE INHIBITING RAF KINASE AND VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTOR, METHOD FOR PREPARING SAME, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND USE THEREOF 삼진제약주식회사 2017-08-10 WO disclosed