Pd-0299685

Pd-0299685

SCHEMBL1923707

CCC[C@@H](C)C[C@@H](CN)CC(=O)O

nearest known ligand 0.63

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 2/20 0.63
ADRA1A P35348 2/20 0.63
CACNB3 P54284 1/20 0.63
CACNA1C Q13936 1/20 0.63
PGR P06401 1/20 0.63
HTR2B P41595 1/20 0.63
CACNA2D2 Q9NY47 1/20 0.63
GABRR1 P24046 2/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.35
GPR84 Q9NQS5 4/20 0.35
GRIK1 P39086 1/20 0.35
SLC1A3 P43003 1/20 0.35
SLC1A2 P43004 1/20 0.35
SLC1A1 P43005 1/20 0.35
GRIK2 Q13002 1/20 0.35
TDP1 Q9NUW8 2/20 0.34
CHRM1 P11229 1/20 0.34
AKR1A1 P14550 1/20 0.34
CHRM3 P20309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pd-0299685 SCHEMBL4382735 1.00 CACNA2D1 (0.63) CACNA2D1ADRA1ACACNB3CACNA1CPGR
Pd-0299685 SCHEMBL119378 1.00 CACNA2D1 (0.63) CACNA2D1ADRA1ACACNB3CACNA1CPGR
Pd-0299685 SCHEMBL588075 1.00 CACNA2D1 (0.63) CACNA2D1ADRA1ACACNB3CACNA1CPGR
Pd-0299685 SCHEMBL3124421 1.00 CACNA2D1 (0.63) CACNA2D1ADRA1ACACNB3CACNA1CPGR
Pd-0299685 SCHEMBL1923704 1.00 CACNA2D1 (0.63) CACNA2D1ADRA1ACACNB3CACNA1CPGR
Pd-0299685 SCHEMBL25912 1.00 CACNA2D1 (0.63) CACNA2D1ADRA1ACACNB3CACNA1CPGR
Pd-0299685 SCHEMBL3123592 0.98 CACNA2D1 (0.61) CACNA2D1ADRA1ACACNB3CACNA1CPGR
Pd-0299685 SCHEMBL3828529 0.98 CACNA2D1 (0.61) CACNA2D1ADRA1ACACNB3CACNA1CPGR
Pd-0299685 SCHEMBL4378882 0.98 CACNA2D1 (0.61) CACNA2D1ADRA1ACACNB3CACNA1CPGR
Pd-0299685 SCHEMBL3828531 0.98 CACNA2D1 (0.61) CACNA2D1ADRA1ACACNB3CACNA1CPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125021-B1 COMBINATION THERAPY OF LOWER URINARY TRACT DISORDERS WITH 2 LIGANDS AND NSAIDS RECORDATI IRELAND LTD (IE) 2011-06-08 EP claimed
EP-1192125-B1 MONO-SUBSTITUTED 3-PROPYL GAMMA-AMINOBUTYRIC ACIDS WARNER LAMBERT CO (US) 2008-12-31 EP claimed
EP-4506001-A2 SUBSTITUTED TETRAHYDROFURANS AS MODULATORS OF SODIUM CHANNELS Vertex Pharmaceuticals Incorporated (US) 2025-02-12 EP disclosed
EP-3651752-B1 CARBOXAMIDES AS MODULATORS OF SODIUM CHANNELS VERTEX PHARMA (US) 2024-11-20 EP disclosed
EP-4069691-B1 SUBSTITUTED TETRAHYDROFURANS AS MODULATORS OF SODIUM CHANNELS VERTEX PHARMA (US) 2024-09-18 EP disclosed
EP-2240467-B1 AMIDE DERIVATIVES AS ION-CHANNEL LIGANDS AND PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING THE SAME EVOTEC AG (DE) 2013-03-20 EP disclosed
EP-1948615-B1 Pyrazole derivatives useful for the treatment of gynaecological diseases PFIZER LTD (GB) 2011-12-14 EP disclosed
EP-2172197-A1 Octanoic acid derivative to treat fibromyalgia and other pains Warner-Lambert Company LLC (US) 2010-04-07 EP disclosed