SCHEMBL19251183

SCHEMBL19251183

O=C1C[C@H]2C1CN2C(=O)OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.52
PSEN1 P49768 2/20 0.50
PSEN2 P49810 2/20 0.50
APH1B Q8WW43 2/20 0.50
NCSTN Q92542 2/20 0.50
APH1A Q96BI3 2/20 0.50
PSENEN Q9NZ42 2/20 0.50
AGTR2 P50052 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
CTRB1 P17538 1/20 0.46
GAA P10253 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24438696 0.84 PREP (0.55) SMN1; SMN2NPC1RAB9ACTRB1
SCHEMBL12458051 0.77 PSEN1 (0.49) HTR2CPSEN1PSEN2APH1BNCSTN
SCHEMBL927563 0.77 PSEN1 (0.49) HTR2CPSEN1PSEN2APH1BNCSTN
SCHEMBL5517082 0.76 HTR2C (0.64) HTR2CPSEN1PSEN2APH1BNCSTN
SCHEMBL5517077 0.76 HTR2C (0.64) HTR2CPSEN1PSEN2APH1BNCSTN
SCHEMBL10053573 0.76 HTR2C (0.64) HTR2CPSEN1PSEN2APH1BNCSTN
SCHEMBL22537068 0.76 HTR2C (0.53) HTR2CPSEN1PSEN2APH1BNCSTN
SCHEMBL1978499 0.76 PSEN1 (0.48) HTR2CPSEN1PSEN2APH1BNCSTN
SCHEMBL21193323 0.76 HTR2C (0.53) HTR2CPSEN1PSEN2APH1BNCSTN
SCHEMBL29278490 0.76 HTR2C (0.53) HTR2CPSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732083-B2 Tricyclic gyrase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-15 US disclosed