SCHEMBL19256853

SCHEMBL19256853

CC1C=CN=C(c2ccsc2)C=C1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 1/20 0.35
HTR2B P41595 1/20 0.35
HTR3A P46098 1/20 0.35
HTR5A P47898 1/20 0.35
CYP2A6 P11509 8/20 0.34
CYP2B6 P20813 3/20 0.33
CYP2E1 P05181 2/20 0.33
ADORA2A P29274 4/20 0.33
ADORA3 P0DMS8 3/20 0.33
ADORA1 P30542 3/20 0.33
ADORA2B P29275 2/20 0.33
KCNH2 Q12809 1/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19257181 0.66 HTR1D (0.34) HTR1DHTR2BHTR3AHTR5ACYP2A6
SCHEMBL18902620 0.63
SCHEMBL2125063 0.61 CYP2A6 (0.72) CYP2A6CYP2B6CYP2E1KCNH2CYP3A4
SCHEMBL3157632 0.60 CYP2A6 (0.41) HTR1DHTR2BHTR3AHTR5ACYP2A6
SCHEMBL22734811 0.58 CYP2A6 (0.52) CYP2A6CYP2B6CYP2E1KCNH2CYP3A4
SCHEMBL29136542 0.58 CYP2A6 (0.59) HTR1DHTR2BHTR3AHTR5ACYP2A6
SCHEMBL2782336 0.57 CYP2A6 (0.58) CYP2A6CYP2B6CYP2E1KCNH2CYP3A4
SCHEMBL18936327 0.57
SCHEMBL20286581 0.57 CYP2A6 (0.34) HTR1DCYP2A6CYP2B6CYP2E1CYP3A4
SCHEMBL27989815 0.57 CYP2A6 (0.74) CYP2A6CYP2B6CYP2E1KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133630-A1 INHIBITOR OF BRUTON'S TYROSINE KINASE 北京盛诺基医药科技有限公司 2017-08-10 WO disclosed