SCHEMBL19257908

SCHEMBL19257908

C[C@@H](CC(N)Cc1ccccc1)C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPI P09923 1/20 0.56
PKM P14618 1/20 0.56
PTGS1 P23219 1/20 0.56
XIAP P98170 1/20 0.56
SLC7A5 Q01650 1/20 0.56
EPHX1 P07099 1/20 0.55
SLC1A3 P43003 2/20 0.53
SLC1A2 P43004 2/20 0.53
SLC1A1 P43005 2/20 0.53
SLC6A2 P23975 2/20 0.52
TAAR1 Q96RJ0 2/20 0.52
MAOA P21397 1/20 0.52
SLC6A4 P31645 1/20 0.52
SLC6A3 Q01959 1/20 0.52
SIGMAR1 Q99720 1/20 0.52
CYP2A6 P11509 1/20 0.52
ADORA2A P29274 1/20 0.52
ADORA1 P30542 1/20 0.52
ENPEP Q07075 2/20 0.52
ANPEP P15144 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16410936 1.00 ALPI (0.56) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL22199422 1.00 ALPI (0.56) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL10063806 1.00 ALPI (0.56) ALPIPKMPTGS1XIAPSLC7A5
Hydrochloric Acid SCHEMBL16278915 0.98 ALPI (0.55) ALPIPKMPTGS1XIAPSLC7A5
Trifluoroacetic Acid SCHEMBL29854324 0.92 ALPI (0.49) ALPIPKMPTGS1XIAPSLC7A5
Trifluoroacetic Acid SCHEMBL28689356 0.92 ALPI (0.49) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL8198670 0.90 MME (0.62) GPR88MMEACE
SCHEMBL1908547 0.90 MME (0.62) GPR88MMEACE
SCHEMBL20580875 0.90 MME (0.62) GPR88MMEACE
SCHEMBL2706785 0.90 MME (0.62) GPR88MMEACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020022892-A1 TUBULYSIN DERIVATIVES AND METHODS FOR PREPARING THE SAME RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-01-30 WO disclosed
WO-2017134547-A1 TUBULYSIN ANALOGS AND METHODS FOR THEIR PREPARATION PFIZER INC. (US) 2017-08-10 WO disclosed