SCHEMBL19265293

SCHEMBL19265293

CNCCn1c(Sc2cc3c(cc2I)OCCO3)nc2c(N)nccc21

nearest known ligand 0.90

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 20/20 0.90
CDC37 Q16543 2/20 0.71
HSP90B1 P14625 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4997743 0.94 HSP90AA1 (1.00) HSP90AA1CDC37HSP90B1
SCHEMBL1743406 0.89 HSP90AA1 (0.90) HSP90AA1CDC37
SCHEMBL2993375 0.89 HSP90AA1 (0.89) HSP90AA1CDC37HSP90B1
SCHEMBL12454183 0.87 HSP90AA1 (0.90) HSP90AA1CDC37HSP90B1
SCHEMBL18431833 0.87 HSP90AA1 (0.90) HSP90AA1CDC37HSP90B1
SCHEMBL18431832 0.87 HSP90AA1 (0.90) HSP90AA1CDC37HSP90B1
SCHEMBL1742677 0.85 HSP90AA1 (1.00) HSP90AA1CDC37HSP90B1
SCHEMBL1743323 0.85 HSP90AA1 (1.00) HSP90AA1CDC37HSP90B1
SCHEMBL4136026 0.84 HSP90AA1 (1.00) HSP90AA1CDC37HSP90B1
SCHEMBL24725170 0.84 HSP90AA1 (0.82) HSP90AA1CDC37HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3709022-A1 USES OF LABELED HSP90 INHIBITORS Sloan-Kettering Institute for Cancer Research (US) 2020-09-16 EP disclosed
EP-3208615-A2 USES OF LABELED HSP90 INHIBITORS Sloan Kettering Institute For Cancer Research (US) 2017-08-23 EP disclosed