SCHEMBL19281131

SCHEMBL19281131

COc1cc(C(=O)N2CCC3(CC2)CC(O)c2ccccc2O3)ccc1C(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACACB O00763 8/20 0.45
MGLL Q99685 1/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
EPHX1 P07099 1/20 0.42
EPHX2 P34913 1/20 0.42
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
USP2 O75604 1/20 0.40
TSHR P16473 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
IDO1 P14902 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19281124 0.87 ACACB (0.46) ACACBKMT2AALDH1A1CYP1A2IDO1
SCHEMBL12695096 0.87 ACACB (0.42) ACACBMGLLMEN1KMT2AEPHX1
SCHEMBL12480905 0.85 ACACB (0.44) ACACBMEN1KMT2AALDH1A1
SCHEMBL19289399 0.84 EPHX2 (0.60) ACACBMGLLEPHX1EPHX2HSP90AA1
SCHEMBL2585266 0.81 ACACB (0.54) ACACBMGLLEPHX1EPHX2
SCHEMBL12695093 0.81 ACACB (0.41) ACACBMGLLMEN1KMT2AEPHX1
SCHEMBL12695166 0.81 ACACB (0.41) ACACBMGLLMEN1KMT2AEPHX1
SCHEMBL19289442 0.81 ACACB (0.41) ACACBMGLLMEN1KMT2AEPHX1
SCHEMBL12481588 0.81 HTT (0.51) MGLLKMT2ATSHRALDH1A1IDO1
SCHEMBL12481302 0.79 ACACB (0.40) ACACBMGLLMEN1KMT2AEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675812-B1 CHROMAN - SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2017-08-30 EP disclosed