SCHEMBL19281152

SCHEMBL19281152

[2H]C([2H])([2H])OCC1CC2(CCN(C(=O)c3ccc(OC(C)C)c(OC)c3)CC2)Oc2cc(F)ccc21

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACACB O00763 5/20 0.39
CYP2D6 P10635 3/20 0.39
ALDH1A1 P00352 2/20 0.38
PKM P14618 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
CCR3 P51677 1/20 0.36
KMT2A Q03164 1/20 0.36
POLB P06746 1/20 0.36
CYP2C19 P33261 1/20 0.36
HPGD P15428 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19281150 0.91 ACACB (0.40) ACACBALDH1A1KDM4EKMT2APOLB
SCHEMBL12480972 0.86 ACACB (0.42) ACACBALDH1A1KDM4EKMT2APOLB
SCHEMBL19289249 0.86 ACACB (0.42) ACACBALDH1A1KDM4EKMT2APOLB
SCHEMBL12695231 0.84 ACACB (0.42) ACACBCYP2D6ALDH1A1PKMKDM4E
SCHEMBL12695071 0.84 CYP2D6 (0.42) ACACBCYP2D6ALDH1A1PKMKDM4E
SCHEMBL12695055 0.82 ACACB (0.41) ACACBALDH1A1KDM4EKMT2APOLB
SCHEMBL12695115 0.82 ACACB (0.41) ACACBCYP2D6ALDH1A1PKMKDM4E
SCHEMBL12480927 0.81 ACACB (0.40) ACACBALDH1A1KDM4EKMT2APOLB
SCHEMBL19281145 0.81 EPHX2 (0.39) ACACBCYP2D6ALDH1A1TSHR
SCHEMBL12695070 0.81 ACACB (0.40) ACACBALDH1A1KDM4EKMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675812-B1 CHROMAN - SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2017-08-30 EP disclosed