SCHEMBL192827

SCHEMBL192827

Clc1cc(Sc2cc(Nc3nc(CCc4ccccc4)cs3)ncc2Br)c(Br)cn1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GCK P35557 7/20 0.42
NOS1 P29475 1/20 0.38
AOC3 Q16853 5/20 0.36
HDAC1 Q13547 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
MAOB P27338 2/20 0.33
SLC2A1 P11166 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
PDE5A O76074 1/20 0.32
PDE1A P54750 1/20 0.32
PDE1B Q01064 1/20 0.32
PDE1C Q14123 1/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL190650 0.90 GCK (0.45) GCKNOS1AOC3HDAC1HDAC6
SCHEMBL12305709 0.85 GCK (0.38) GCKNOS1AOC3HDAC1HDAC6
SCHEMBL191831 0.84 GCK (0.41) GCKNOS1AOC3
SCHEMBL191232 0.82 GCK (0.41) GCKNOS1AOC3MEN1NPC1
SCHEMBL191869 0.82 GCK (0.44) GCKNOS1AOC3MAOBGAA
SCHEMBL192067 0.82 GCK (0.44) GCKNOS1AOC3HDAC1HDAC6
SCHEMBL190783 0.82 GCK (0.40) GCKNOS1AOC3HDAC1HDAC6
SCHEMBL191596 0.81 GCK (0.44) GCKNOS1AOC3HDAC1HDAC6
SCHEMBL192244 0.81 GCK (0.44) GCKNOS1AOC3HDAC1HDAC6
Hydrochloric Acid SCHEMBL191165 0.80 GCK (0.43) GCKNOS1AOC3HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1986645-B1 GLUCOKINASE ACTIVATORS ARRAY BIOPHARMA INC (US) 2012-01-04 EP disclosed