SCHEMBL19288129

SCHEMBL19288129

COCCOCC(=O)c1ccc(NS(=O)(=O)c2cc(-c3ccc4c(c3)CCO4)c(Cl)s2)cc1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 3/20 0.55
FABP4 P15090 3/20 0.38
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
PKM P14618 2/20 0.36
MAPT P10636 1/20 0.36
IDH1 O75874 1/20 0.36
POLQ O75417 1/20 0.36
PKLR P30613 1/20 0.35
BRD4 O60885 1/20 0.35
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15055421 0.90 PFKFB3 (0.57) PFKFB3FABP4HDAC3HDAC4HDAC1
SCHEMBL15055585 0.87 PFKFB3 (0.62) PFKFB3FABP4HDAC3HDAC4HDAC1
SCHEMBL9997131 0.84 PFKFB3 (0.76) PFKFB3FABP4PKMMAPTIDH1
SCHEMBL30268499 0.84 PFKFB3 (0.76) PFKFB3FABP4PKMMAPTIDH1
SCHEMBL15080000 0.78 PFKFB3 (0.52) PFKFB3FABP4PKMMAPTSMN1; SMN2
SCHEMBL15058769 0.78 PFKFB3 (0.73) PFKFB3PKMMAPTTSHRSMN1; SMN2
SCHEMBL15080044 0.76 PFKFB3 (0.49) PFKFB3FABP4HDAC3HDAC4HDAC1
Trifluoroacetic Acid SCHEMBL16393839 0.75 PFKFB3 (0.49) PFKFB3FABP4PKM
SCHEMBL15059401 0.75 PFKFB3 (0.48) PFKFB3FABP4HDAC3HDAC4HDAC1
SCHEMBL15058582 0.74 PFKFB3 (0.82) PFKFB3PKMMAPTTSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2794009-B1 BISARYLSULFONAMIDES USEFUL IN THE TREATMENT OF INFLAMMATION AND CANCER KANCERA AB (SE) 2017-08-30 EP disclosed