SCHEMBL19320669

SCHEMBL19320669

COC(=O)c1cnc(Nc2cc([N+](=O)[O-])c(N(C)CCN(C)C)cc2OC)nc1-n1ccc2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.55
ERBB2 P04626 1/20 0.45
ERBB3 P21860 1/20 0.45
ERBB4 Q15303 1/20 0.45
KCNH2 Q12809 2/20 0.43
INSR P06213 1/20 0.43
IGF1R P08069 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19103306 0.94 EGFR (0.60) EGFRERBB2ERBB3ERBB4
SCHEMBL22510210 0.92 EGFR (0.56) EGFRERBB4INSRIGF1R
SCHEMBL29464116 0.89 EGFR (0.49) EGFRKCNH2INSRIGF1R
SCHEMBL29464132 0.87 EGFR (0.49) EGFRKCNH2INSRIGF1R
SCHEMBL17385193 0.86 EGFR (0.76) EGFR
SCHEMBL17384772 0.86 EGFR (0.51) EGFRERBB4INSRIGF1R
SCHEMBL19100929 0.84 EGFR (0.54) EGFRERBB2ERBB3KCNH2INSR
SCHEMBL17385199 0.82 EGFR (0.61) EGFRERBB2ERBB3ERBB4KCNH2
SCHEMBL19103377 0.82 EGFR (0.63) EGFRERBB2ERBB3ERBB4
SCHEMBL17373069 0.82 EGFR (0.74) EGFRERBB2ERBB3ERBB4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170253594-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-09-07 US disclosed
US-20170253594-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-09-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170253594-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ERBB2, EGFR, ERBB3 EGFR 2/4885ERBB2 1/4885ERBB3 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.